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Search Results for " nachrs partial agonist "

6

Compounds

Cat No. Product Name Synonyms Targets
T4246 Varenicline dihydrochloride AChR
Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.
T2285 Encenicline hydrochloride EVP-6124 (hydrochloride),EVP-6124 hydrochloride AChR
Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).
T40431 Anabaseine
Anabaseine is a non-selective nicotinic agonist that stimulates all alpha-7 subtypes of AChRs, with a preference for skeletal muscle and brain. Additionally, it acts as a weak partial agonist at alpha-4 beta-2 nAChRs.
T9450 NS3861 fumarate
NS3861 fumarate is an agonist of nicotinic acetylcholine receptors (nAChRs). NS3861 fumarate is a partial agonist at α3β4 nAChR and binds with high affinity to heteromeric α3β4 nAChR. The binding Ki values of 0.62, 25, 7...
T16563 Pozanicline ABT-089 AChR
Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction. Pozanicline selectively activate neuronal nicotinic acetylcholine...
T4246L Varenicline
Varenicline (CP 526555), a cytisine-based nicotinic ligand, is a potent partial agonist for the α4β2 nicotinic acetylcholine receptor (nAChR) with an EC50 value of 2.3 μM and acts as a full agonist for α7 and α3β4 nAChRs...
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